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Patient Characteristics Associated with Tuberculosis Treatment Default: A Cohort Study in a High-Incidence Area of Lima, Peru
(Public Library of Science, 2015)
BACKGROUND: Although tuberculosis (TB) is usually curable with antibiotics, poor adherence to medication can lead to increased transmission, drug resistance, and death. Prior research has shown several factors to be ...
Dihydro-β-agarofuran sesquiterpenes isolated from Celastrus vulcanicola as potential anti-Mycobacterium tuberculosis multidrug-resistant agents
(Elsevier, 2011)
In the present study, we report four new dihydro-β-agarofuran sesquiterpenes (1-4), which were isolated from the leaves of Celastrus vulcanicola, in addition to five derivatives (5-9). Their stereostructures were elucidated ...
Antibacterial, antifungal and antileishmanial activities of indolone-N-oxide derivatives
(Springer, 2012)
An alarming increase in microbial resistance to traditional drugs and classical pharmacophores has spurred the search for new antimicrobial compounds. Indolone-N-oxides (INODs) possess a redox pharmacophore with promising, ...
Fluoromicobacteriófagos para el screening rápido de alto rendimiento de drogas antituberculosasFluoromycobacteriophages for rapid high-throughput screening of antitubercular drugs
(2018-12-11)
La Tuberculosis (TB) es una enfermedad infecciosa que constituye uno de los mayores problemas sanitarios a nivel mundial. Millones de personas contraen la enfermedad, tanto que a partir de 2015 se localizó dentro de las ...
Diseño in silico, síntesis y efecto en la actividad Ca2+ -ATPasa de CtpF de los compuestos derivados del núcleo pirrolo[1,2- a]quinoxalinas con potencial antimicobacteriano
(Universidad Nacional de ColombiaBogotá - Ciencias - Maestría en Ciencias - BioquímicaDepartamento de QuímicaFacultad de CienciasBogotá, ColombiaUniversidad Nacional de Colombia - Sede Bogotá, 2021)
La Ca2+-ATPasa tipo P de CtpF de Mycobacterium tuberculosis (Mtb), es un transportador de membrana fundamental en la homeóstasis iónica y la viabilidad celular de la micobacteria; posee un sitio de unión cuya interacción ...
Análisis de la distribución de flujo metabólico para la síntesis de ácido micólico en Mycobacterium tuberculosis, aislado clínico UT205
(Escuela de biocienciasUniversidad Nacional de Colombia - Sede Medellín, 2017-06-16)
[Title: Metabolic flux analysis of mycolic acid pathway, Mycobacterium tuberculosis clinical isolate UT205]
Every year in Colombia, there are more than eleven thousand new cases of tuberculosis, indicating that this disease ...