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N-acylation of lactams derived from natural 2-benzoxazolinones and 1,4-benzoxazin-3-ones
(Sociedad Chilena de Quimica, 1999)
The N-acylation reaction of a series of lactams of biological interest, derived from 2-benzoxazolinones and 1,4-benzoxazin-3-one, with acetic anhydride has been studied. The reaction yields show the same tendency as that ...
Heck arylations of N-acyl-3-pyrroline and N-acyl-1,2,5,6-tetrahydropyridine with aryldiazonium salts. Short syntheses of aryl gamma- and delta-lactams, baclofen, homobaclofen and analogues
(Pergamon-elsevier Science LtdOxfordInglaterra, 2002)
Synthesis of (5R)-4-Methyl-5-phenyl-1,3,4-oxadiazinan-2-one and some N-acyl derivatives from (R)-phenylglycine
(Georg Thieme Verlag KgStuttgartAlemanha, 2005)
1,n-diamines. Part 2: Synthesis of acyclic and heterocyclic N-arylputrescine derivatives
(Pergamon-Elsevier Science Ltd, 2011-04)
In the present Letter we report the use of N-arylputrescines as synthetic intermediates for the preparation of N-acyl-N′-aryltetramethylenediamines 3 and related seven-membered heterocyclic amidines 4. Compounds 1 were ...
On the cytotoxic activity of Pd(II) complexes of N,N-disubstituted-N′-acyl thioureas
(ElsevierPhiladelphia, 2014-05)
The rational design of anticancer drugs is one of the most promising strategies for increasing their cytotoxicity and for minimizing their toxicity. Manipulation of the structure of ligands or of complexes represents a ...
n-3 LCPUFA in the reversal of hepatic steatosis: the role of ACOX and CAT-1
(2016)
The aim of this study was to investigate the roles of the Acyl co-enzyme A oxidase (ACOX), carnitine acyl transferase I (CAT-1) and activating protein 1 (AP-1) in the reversal of hepatic steatosis with dietary change and ...