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El pretratamiento agudo y subcrónico con fármacos anticonvulsivantes modifica las crisis generalizadas inducidas por el pentilenetetrazol en el ratón.
(2012-11-30)
Objetivo: El incremento en el contenido de GABA cerebral o la administración de un agente GABA-mimético se emplea
como un tratamiento antiepiléptico eficaz. Sin embargo, se sugiere que el empleo de fármacos que alteran ...
Anticonvulsant and GABA uptake inhibition properties of venom fractions from the spiders Parawixia bistriata and Scaptocosa raptoria
(Swets Zeitlinger Publishers, 2002-09-01)
In this article we describe an in vivo anticonvulsant effect from denatured crude venom and partially isolated fractions from two spiders: Parawixia bistriata and Scaptocosa raptoria. Intracerebroventricular injections of ...
Avaliação do efeito do composto MPMT-OX sobre neurotransmissão e comportamento convulsivo em Caenorhabditis elegans
(Universidade Federal de Santa MariaBrasilBioquímicaUFSMPrograma de Pós-Graduação em Ciências Biológicas: Bioquímica ToxicológicaCentro de Ciências Naturais e Exatas, 2017-03-06)
Epilepsy is characterized as an increased predisposition of the brain to generate recurrent seizures, which represent the effects of abnormal, excessive and hypersynchronous electrical discharges of cortical neurons. ...
Efeito da administração oral de aflatoxina B1 nas convulsões induzidas em ratos
(Universidade Federal de Santa MariaBRFarmacologiaUFSMPrograma de Pós-Graduação em Farmacologia, 2014-08-14)
Aflatoxins are produced by Aspergillus flavus fungi, mainly A. parasiticus and A. nomius. Aflatoxin B1 (AFB1) is the most common and highly toxic mycotoxin, presents carcinogenic, mutagenic and teratogenic effects. This ...
N,N′-Dicyclohexylsulfamide and N,N′-diphenethylsulfamide are anticonvulsant sulfamides with affinity for the benzodiazepine binding site of the GABAA receptor and anxiolytic activity in mice
(Elsevier Inc, 2012-01)
A set of sulfamides designed, synthesized and evaluated against maximal electroshock seizure (MES) and pentilenetetrazol (PTZ) tests with promising results, were tested for their affinity for the benzodiazepine binding ...