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Ausência de efeito antinociceptivo decorrente da administração intravenosa de crotalfina em comparação com morfina, U50-488H ou fenilbutazona em equinos submetidos à estimulação térmica da pele íntegra
(Universidade Federal de Santa Maria (UFSM), 2013-04-01)
Crotalfina é um novo peptídeo analgésico que atua em receptores opioides kappa e delta promovendo potente analgesia em ratos submetidos a modelos de dor inflamatória, neuropática ou oncológica. Talvez a crotalfina possa ...
Influência do consumo de gordura interesterificada nos períodos iniciais do desenvolvimento sobre parâmetros de adição por morfina em ratas
(Universidade Federal de Santa MariaBrasilFarmacologiaUFSMPrograma de Pós-Graduação em FarmacologiaCentro de Ciências da Saúde, 2017-02-17)
There is a high consumption of processed foods with interesterified fat (IF), which has
replaced trans fat, given that it has shown harmful effects on health. Morphine is an opioid
drug, widely used to alleviate acute ...
Restraint stress enhances alcohol intake in adolescent female rats but reduces alcohol intake in adolescent male and adult female rats
(Elsevier Science, 2017-08-10)
Adolescents may be more sensitive to stress-induced alcohol drinking than adults, which would explain the higher prevalence of alcohol abuse and dependence in late adolescence than in adulthood. The present study analyzed ...
Ausência de efeito antinociceptivo decorrente da administração intravenosa de crotalfina em comparação com morfina, U50-488H ou fenilbutazona em equinos submetidos à estimulação térmica da pele íntegra
(Universidade Federal de Santa Maria (UFSM), 2014)
Behavioral effects of acute stimulation of kappa-opioid receptors during lactation
(PERGAMON-ELSEVIER SCIENCE LTD, 2008)
The behavioral effects of the K-opioid receptor agonist U69593 were examined in lactating rats. On day 5 of lactation, animals were treated with 0.1 mg/kg of U69593 to determine whether it influences general activity and ...
Usos terapéuticos potenciales de los antagonistas opioides: Fisiopatología y evidencia preclínica
(Universidad Nacional de Colombia - Sede Bogotá - Facultad de Ciencias - Departamento de Farmacia, 2015-09-01)
El sistema opioide, del cual forman parte los péptidos opioides endógenos y sus receptores (Miu, Kappa, delta y ORL), tiene un papel importante en la fisiología de diferentes sistemas. Existe una creciente evidencia de su ...
Peripheral Sensitization Increases Opioid Receptor Expression And Activation By Crotalphine In Rats
(Public Library of Science, 2014)
Stimulation of peripheral Kappa opioid receptors inhibits inflammatory hyperalgesia via activation of the PI3K gamma/AKT/nNOS/NO signaling pathway
(BIOMED CENTRAL LTDLONDON, 2012)
Background: In addition to their central effects, opioids cause peripheral analgesia. There is evidence showing that peripheral activation of kappa opioid receptors (KORs) inhibits inflammatory pain. Moreover, peripheral ...