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Synthesis, binding assays, cytotoxic activity and docking studies of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid receptor
(Elsevier, 2016)
Herein we report the design, synthesis, bioinformatic and biological studies of benzimidazole and benzothiophene derivatives as new cannabinoid receptor ligands. To test the hypothesis that the lack of a hydrogen bond ...
Síntese e aplicação de nanofiltro contendo nanotubos de carbono na retenção de contaminantes em água
(Universidade Federal de Santa MariaBREngenharia AgrícolaUFSMPrograma de Pós-Graduação em Engenharia Agrícola, 2015-06-05)
This work aimed to use Multiple Walls Nanotubes (MWNT) in order to synthesize a nanofilter to remove water contaminants and to test the nanofilter manufactured in removing Benzothiophene and pesticides present in water. ...
Synthesis, binding assays, cytotoxic activity and docking studies of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid receptor
(2016)
Herein we report the design, synthesis, bioinformatic and biological studies of benzimidazole and benzothiophene derivatives as new cannabinoid receptor ligands. To test the hypothesis that the lack of a hydrogen bond ...
Synthesis of benzo[b]thiophene carboxamides connected to 4-arylpiperazines through a benzylic spacer: Potential Ligands with 5-HT1A binding affinity
(TAYLOR & FRANCIS INC, 2007)
New benzothiophene arylpiperazine derivatives 8 (a-f) were synthesized as potential serotoninergic agents with 5-HT1A receptor affinity. Preparation of the derivatives was performed by treating N-[2-(chloromethyl)phenyl] ...
Synthesis, binding assays, cytotoxic activity and docking studies of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid receptor
(2016)
Herein we report the design, synthesis, bioinformatic and biological studies of benzimidazole and benzothiophene derivatives as new cannabinoid receptor ligands. To test the hypothesis that the lack of a hydrogen bond ...
Self Diffusivity of n-Dodecane and Benzothiophene in ZSM-5 Zeolites: Its Significance for a New Catalytic Light Diesel Desulfurization Process
(Berkeley Electronic Press, 2016-06-13)
This study provides theoretical support to a recent promising ZSM5 catalyst used for the selective desulfurization of light diesel type compounds (Al-Bogami and de Lasa 2013; Al-Bogami, Moreira, and de Lasa 2013). With ...
Versatile one-pot synthesis of benzo-fused thiacycles by copper catalysis
(Royal Society of Chemistry, 2017-04)
A novel, one-pot synthesis of structurally diverse benzo-fused thiacycles via a Cu-catalysed intermolecular C?S coupling/cyclisation tandem process, employing the same catalytic system, has been developed. Thus, ...
Solvent-free microwave synthesis of 3-(4-benzo[b]-thiophene-2-carbonyl)-1-piperazinyl-1-benzo[b]thiophen-2-YL-1-propanones. New hetero bis-ligands with potential 5-HT1A serotonergic activity
(2008)
A novel series of 2-benzothiophenealkylpiperazine derivatives 11 (a-d) with potential affinity at 5-HT1A serotonin receptors have been synthesized via solvent-free, microwave-promoted Michael addition of benzo[b]thiophene ...
Solvent-free microwave synthesis of 3-(4-benzo[b]thiophene-2-carbonyl)-1-piperazinyl-1-benzo[b]thiophen-2-yl-1-propanones. New hetero bis-ligands with potential 5-HT1A serotonergic activity
(PERGAMON-ELSEVIER SCIENCE LTD, 2008)
A novel series of 2-benzothiophenealkylpiperazine derivatives 11 (a-d) with potential affinity at 5-HT1A serotonin receptors have been synthesized via solvent-free, microwave-promoted Michael addition of benzo[b]thiophene ...