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Practical synthesis of chiral beta-telluro amines by ring-opening reaction of aziridines

VARGAS, Fabricio; COMASSETO, Joao V. (ELSEVIER SCIENCE SA, 2009)

A set of chiral beta-tellurium amines and their selenium and sulfur-containing derivatives have been efficiently synthesized in good to excellent yields via the ring-opening reaction of chiral aziridines by chalcogen ...

Catalytic stereoselective alkene aziridination with sulfonimidamides

Robert-Peillard, Fabien; Di Chenna, Pablo Hector; Liang, Chungen; Lescot, Camille; Collet, Florence; Dodd, Robert H.; Dauban, Philippe (Pergamon-Elsevier Science Ltd, 2010-06)

Diastereoselective copper-catalyzed alkene aziridination has been investigated using chiral nitrenes generated from sulfonimidamides in the presence of an iodine(III) oxidant. Starting from a stoichiometric amount of the ...

Theoretical aspects of binary and ternary complexes of aziridine???ammonia ruled by hydrogen bond strength

Oliveira, Boaz G.; Ara??jo, Regiane C. M. U. (2012)

Aziridination of 11-pregnene-3,20-dione using PhI=N-Ses

Di Chenna, Pablo Hector; Dauban, Philippe; Ghini, Alberto Antonio; Burton, Gerardo; Dodd, Robert H. (Pergamon-Elsevier Science Ltd, 2000-09)

The copper-catalyzed reaction of [N-(Ses)imino]phenyliodinane with 11-pregnene-3,20-dione gave the corresponding aziridine in 53% yield. The Ses protecting group could be conveniently removed using the TASF reagent. ...

Intramolecular Phl=O mediated copper-catalyzed aziridination of unsaturated sulfamates: A new direct access to polysubstituted amines from simple homoallylic alcohols

Duran, Fernando Javier; Leman, Loïc; Ghini, Alberto Antonio; Burton, Gerardo; Dauban, Philippe; Dodd, Robert H. (American Chemical Society, 2002-07)

(Matrix presented) Olefinic sulfamates derived from primary and secondary alcohols undergo intramolecular copper-catalyzed aziridination in the presence of iodosylbenzene to afford novel bicyclic fused aziridines. The ...

Theoretical aspects of binary and ternary complexes of aziridine⋯ammonia ruled by hydrogen bond strength

Oliveira, Boaz G.; Araújo, Regiane C. M. U.; Oliveira, Boaz G.; Araújo, Regiane C. M. U. (Brasil, 2012)

B3LYP calculations, ChelpG atomic charges, and quantum theory of atoms in molecules (QTAIM) integrations were used to investigate the binary (1:1) and ternary (1:2) hydrogen-bonded complexes formed by aziridine (1) and ...

Aziridine-2,3-dicarboxylate inhibitors targeting the major cysteine protease of Trypanosoma brucei as lead trypanocidal agents

Vicik, Radim; Hoerr, Verena; Glaser, Melanie; Schultheis, Martina; Hansell, Elizabeth; McKerrow, James H.; Holzgrabe, Ulrike; Caffrey, Conor R.; Ponte-Sucre, Alicia; Moll, Heidrun; Stich, August; Schirmeister, Tanja (2012)

Aziridine-2,3-Dicarboxylates, Peptidomimetic Cysteine Protease Inhibitors with Antileishmanial Activity

Ponte-Sucre, Alicia; Vicik, Radim; Schultheis, Martina; Schirmeister, Tanja; Moll, Heidrun (2012)

Synthesis of a Trihydroxylated Aminoazepane from D-Glucitol by an Intramolecular Aziridine Ring Opening

Valle, MS; Braga, RM (Georg Thieme Verlag KgStuttgartAlemanha, 2008)

Development of a New Antileishmanial Aziridine-2,3-Dicarboxylate-Based Inhibitor with High Selectivity for Parasite Cysteine Proteases.

Schad, Croline; Baum, Ulrike; Frank, Benjamin; Dietzel, Uwe; Mattern, Felix; Gomes, Carlos; Ponte-Sucre, Alicia; Moll, Heidrun; Schurigt, Uta; Schirmeister, Tanja (2016)

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