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A novel physiological property of snake bradykinin-potentiating peptides-Reversion of MK-801 inhibition of nicotinic acetylcholine receptors
(ELSEVIER SCIENCE INC, 2008)
The first naturally occurring angiotensin-converting enzyme (ACE) inhibitors described are pyroglutamyl proline-rich oligopeptides, found in the venom of the viper Bothrops jararaca, and named as bradykinin-potentiating ...
Avaliação do papel da D-serina na modulação da resposta de inibição por pré-pulso do reflexo de sobressalto acústico em um modelo animal de esquizofrenia: ratos wistar machos tratados agudamente com MK-801
(Universidade Federal de São Paulo (UNIFESP), 2021)
Schizophrenia is a mental disorder that affects approximately 1% of the world population, being a chronic and debilitating pathology. One of the neurochemical hypotheses related to schizophrenia is the existence of a ...
Effects of MK-801 and amphetamine treatments on allergic lung inflammatory response in mice
(Elsevier ScienceAmsterdam, 2013-08-16)
Glutamate acts as a neurotransmitter within the Central Nervous System (CNS) and modifies immune cell activity. In lymphocytes, NMDA glutamate receptors regulate intracellular calcium, the production of reactive oxygen ...
Avaliação do potencial neuroprotetor de fármacos antipsicóticos em alterações bioquímicas, moleculares e comportamentais induzidas por antagonista de receptor NMDA (MK-801) em peixe zebra (Danio rerio)
(Pontifícia Universidade Católica do Rio Grande do SulPorto Alegre, 2011)
Schizophrenia is a severe mental illness characterized by positive and negative symptoms and cognitive deficits. This pathology is still poorly understood. Reduction of glutamatergic neurotransmission by NMDA receptor ...
Avaliação do potencial neuroprotetor de fármacos antipsicóticos em alterações bioquímicas, moleculares e comportamentais induzidas por antagonista de receptor NMDA (MK-801) em peixe zebra (Danio rerio)
(Pontifícia Universidade Católica do Rio Grande do SulPorto Alegre, 2011)
Schizophrenia is a severe mental illness characterized by positive and negative symptoms and cognitive deficits. This pathology is still poorly understood. Reduction of glutamatergic neurotransmission by NMDA receptor ...
Efeito do monossialogangliosídeo GM1 sobre as alterações comportamentais, euroquímicas e eletrográficas induzidas pelo ácido glutárico e nas defesas antioxidantes no SNC de ratos
(Universidade Federal de Santa MariaBRBioquímicaUFSMPrograma de Pós-Graduação em Ciências Biológicas: Bioquímica Toxicológica, 2006-05-12)
Monosialoganglioside (GM1) is a component of most cell membranes and is thought to play a role in development, recognition and cellular differentiation. Furthermore, GM1 is a neuroprotective agent that has been reported ...
Compostos 1,2 e 1,4-dicarboxílicos atuam sobre o sistema glutamatérgico e o comportamento de ratos e camundongos
(Universidade Federal de Santa MariaBRBioquímicaUFSMPrograma de Pós-Graduação em Ciências Biológicas: Bioquímica Toxicológica, 2005-07-27)
Glutamatergic receptors are targets for many L-glutamate structure analogues, which cause neurotoxicity. This study investigated the actions of two dicarboxylic compounds, the first had cyclic framework and rigid structure, ...
Electrophysiological effects of guanosine and MK-801 in a quinolinic acid-induced seizure model
(2010)
Quinolinic acid (QA) is an N-methyl-D-aspartate receptor agonist that also promotes glutamate release and
inhibits glutamate uptake by astrocytes. QA is used in experimental models of seizures studying the effects ...
Sucinato melhora a memória da tarefa de medo condicionado em ratos
(Universidade Federal de Santa MariaBRBioquímicaUFSMPrograma de Pós-Graduação em Ciências Biológicas: Bioquímica Toxicológica, 2007-07-03)
Succinate is a dicarboxylic acid that accumulates due to succinate dehydrogenase inhibition. This dicarboxylic acid has a biphasic effect on neural activity in vitro that seems to be
mediated by N-methyl-D-aspartate (NMDA) ...
Caracterização Farmacológica da Inibição Pré-Pulso ("Prepulse Inhibition of Startle") na Linhagem SHR (Spontaneously Hypertensive Rats): Possíveis Implicações para Transtornos Psiquiátricos
(Universidade Federal de São Paulo (UNIFESP), 2009-04-29)
Deficits in an operational measure of sensorimotor gating - the prepulse inhibition of startle (PPI) - is presented in psychiatric disorders such as schizophrenia, bipolar disorder, and attention deficit/hyperactivity ...