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Panax ginseng metabolite (GIM-1) modulates the effects of monobutyl phthalate (MBP) on the GPR30/GPER1 canonical pathway in human Sertoli cells
(2020-09-01)
This study was performed to evaluate the effect of monobutyl phthalate (MBP) on GPR30-activated pathways in Sertoli cells. Additionally, we tested if GIM-1 (Panax ginseng metabolite) modulates MBP action. Human Sertoli ...
Raloxifene decreases cell viability and migratory potential in prostate cancer cells (LNCaP) with GPR30/GPER1 involvement
(2019-07-01)
Objectives: This study evaluated raloxifene (ral) effects on LNCaP prostate tumour cells modulating the activity of GPER1/GPR30 receptors. Methods: LNCaP cells were submitted for 40/120 min and 12 h to the following ...
Continuous Exposure of Breast Cancer Cells to Tamoxifen Upregulates GPER-1 and Increases Cell Proliferation
(FRONTIERS MEDIA SA, 2020)
Possible role of phytoestrogens in breast cancer via GPER-1/GPR30 signaling
(2018-12-01)
Estrogens generated within endocrine organs and the reproductive system act as ligands for at least three types of estrogen receptors. Estrogen receptors α (ERα) and β (ERβ) belong to the so-called classical family of ...
Participación del receptor de estrógenos acoplado a proteína G (GPER/GPR30) en los efectos no genómicos de aldosterona en el corazón
(2019-03-06)
Los receptores acoplados a proteína G (GPCRs) codifican una amplia variedad de respuestas, como las que se dan a diversos procesos autócrinos, parácrinos y endócrinos. El receptor de estrógenos acoplado a proteína G (GPER) ...
Caracterização dos efeitos celulares do Mono-N-butil-ftalato (MBP) mediados pela via estrogênica não-genômica ativada por GPER1 (GPR30) em células tumorais prostáticas humanasCharacterization of the cellular effects of the mono-N-butyl phthalate (MBP) mediated by non-genomic estrogen pathway activated by GPR30 in human prostate tumor cells
(Universidade Estadual Paulista (Unesp), 2016)
Caracterização dos efeitos celulares do Mono-N-butil-ftalato (MBP) mediados pela via estrogênica não-genômica ativada por GPER1 (GPR30) em células tumorais prostáticas humanas
(Universidade Estadual Paulista (Unesp), 2016-03-04)
The mono-n-butyl phthalate (MBP) is the active metabolite of di-n-butyl phthalate (DBP), a plasticizer commonly used for industrial products, including medical devices, flexible plastics and cosmetics, has been described ...
Caracterização dos efeitos celulares do Mono-N-butil-ftalato (MBP) mediados pela via estrogênica não-genômica ativada por GPER1 (GPR30) em células tumorais prostáticas humanas
(Universidade Estadual Paulista (UNESP), 2016)