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Identification of the potential biological target of N-benzenesulfonyl-1,2,3,4-tetrahydroquinoline compounds active against gram-positive and gram-negative bacteria
(Adenine Press, 2019-06-23)
The development of new antibiotics with activity towards a broad spectrum of bacteria, including multiresistant strains, is a very important topic for global public health. As part of previous works, N-benzenesulfonyl-1, ...
Evaluation of antibacterial activity and reactive species generation of N-benzenesulfonyl derivatives of heterocycles
(Pharmaceutical Soc Japan, 2016-01)
Two N-benzenesulfonyl (BS) derivatives of 1,2,3,4-tetrahydroquinoline (THQ) were designed, prepared,and screened for antibacterial activity. This approach was based on combining the two privileged structures,BS and THQ, ...
Nuevas formas sólidas de compuestos con actividad antiparasitaria : preparación y caracterización
(2021-10-01)
Resumen Las enfermedades parasitarias siguen siendo una de las principales preocupaciones para la salud pública de los países en desarrollo. Entre ellas, las causadas por protozoos tienen un gran impacto porque han resurgido ...
Design, synthesis and 3-d characterization of 1-benzenesulfonyl-1,2,3,4-tetrahydroquinolines as lead scaffold for antiparasitic drug
(Bentham Science Publishers, 2010-10)
Ten 1-benzenesulfonyl-1,2,3,4-tetrahydroquinoline (BSTHQ) were synthesized and characterized and their antiprotozoal activities were investigated. This small library was designed by combining two chemical moieties that are ...