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Design, synthesis and 3-d characterization of 1-benzenesulfonyl-1,2,3,4-tetrahydroquinolines as lead scaffold for antiparasitic drug
(Bentham Science Publishers, 2010-10)
Ten 1-benzenesulfonyl-1,2,3,4-tetrahydroquinoline (BSTHQ) were synthesized and characterized and their antiprotozoal activities were investigated. This small library was designed by combining two chemical moieties that are ...
SAR analysis of new dual targeting fluoroquinolones. Implications of the benzenesulfonyl group
(Bentham Science Publishers, 2012-05)
When a benzenesulfonyl moiety (BS) was bound to the N-piperazinyl ring of antibacterial fluoroquinolones (AMFQs) norfloxacin (NOR) or ciprofloxacin (CIP), the resulting benzenesulfonyl-fluoroquinolone (BSFQs) analogs showed ...
X-ray, DFT, FTIR and thermal study of the antimicrobial N-benzenesulfonyl-1H-1,2,3-benzotriazole
(Elsevier Science, 2018-03)
N-benzenesulfonyl-1H-1,2,3-benzotriazole (NBSBZT) is a compound with significant trypanocidal and bactericidal activities, which we reported previously. In this work a combined experimental and theoretical study of its ...
Novos ligantes e complexos de Sn(IV) com potencial atividade biológica: avaliação da atividade antimicrobiana e estudos cristalográficos
(Universidade Federal de Minas GeraisUFMG, 2018-07-30)
In this work, we present structural variations of compounds that have biological activity reported in the literature through the insertion of R-benzenesulfonyl and isoxazole groups, as well as the complexation of some of ...
THE CATHODIC CLEAVAGE OF THE NITROBENZENESULFONYL GROUP FROM ALIPHATIC-AMINES IN N,N-DIMETHYLFORMAMIDE
(Elsevier B.V., 1991-08-26)
The reduction of benzenesulfonyl derivatives of n-butylamine and N,N-di-n-butylamine with nitro substituents at the 2, 3 and 4 positions of the phenyl ring in N,N-dimethylformamide is reported. The N,N-di-n-butyl-4- and ...
THE CATHODIC CLEAVAGE OF THE NITROBENZENESULFONYL GROUP FROM ALIPHATIC-AMINES IN N,N-DIMETHYLFORMAMIDE
(Elsevier B.V., 1991-08-26)
The reduction of benzenesulfonyl derivatives of n-butylamine and N,N-di-n-butylamine with nitro substituents at the 2, 3 and 4 positions of the phenyl ring in N,N-dimethylformamide is reported. The N,N-di-n-butyl-4- and ...
Síntesis y caracterización de compuestos híbridos del tipo pirimido-sulfonamida con potencial actividad antibacteriana
(Universidad de Ciencias Aplicadas y AmbientalesFacultad de CienciasBogotá, 2023)
En este trabajo se presentan los estudios de acoplamiento molecular de una serie de sistemas híbridos del tipo pirimido-sulfonamida con la proteína dihidropteroato sintasa, así como su comparación con los resultados obtenidos ...