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Muerte celular de fibroblastos y miofibroblastos cardiacos neonatos por sobre-expresión de los receptores tipo 1 y 2 de angiotensina II
(Universidad de ChilePrograma Cybertesis, 2006)
Fibroblastos y miofibroblastos cardiacos son elementos claves en el desarrollo del remodelamiento cardiaco después de un infarto agudo al miocardio. Una regulación controlada en el crecimiento de la población de fibroblastos ...
Translocator protein (18 kDa) mediates the pro-growth effects of diazepam on Ehrlich tumor cells in vivo
(Amsterdam, 2010)
The Translocator Protein (TSPO), previously known as the peripheral-type benzodiazepine receptor, is a ubiquitous drug- and cholesterol-binding protein that is up regulated in several types of cancer cells. TSPO drug ligands ...
Effect of leuprolide and cetrorelix on cell growth, apoptosis, and GnRH receptor expression in primary cell cultures from human prostate carcinoma
(TAYLOR & FRANCIS INC, 2006-05)
Contradictory data have been reported regarding the effect of GnRH agonists and antagonists on cell growth and survival, using prostate cancer-derived cell lines expressing either endogenous or exogenous GnRH receptors. ...
Avaliação dos efeitos cardiovasculares do novo agonista do receptor MAS, CGEN 856S
(Universidade Federal de Minas GeraisUFMG, 2011-05-30)
The increasing evidence of the beneficial effects of Angiotensin-(1-7) [Ang-(1- 7)] through the activation of its receptor Mas, as vasodilation, antiarrhythmogenesis, antitrombogenesis, antifibrogenesis, improvement of ...
Differential antagonism by conotoxin p-TIA of contractions mediated by distinct alpha(1)-adrenoceptor subtypes in rat vas deferens, spleen and aorta
(Elsevier B.V., 2005-01-31)
The ability of the conotoxin p-TIA, a 19-amino acid peptide isolated from the marine snail Conus tulipa, to antagonize contractions induced by noradrenaline through activation of alpha(1A)-adrenoceptors in rat vas deferens, ...
Differential antagonism by conotoxin p-TIA of contractions mediated by distinct alpha(1)-adrenoceptor subtypes in rat vas deferens, spleen and aorta
(Elsevier B.V., 2005-01-31)
The ability of the conotoxin p-TIA, a 19-amino acid peptide isolated from the marine snail Conus tulipa, to antagonize contractions induced by noradrenaline through activation of alpha(1A)-adrenoceptors in rat vas deferens, ...
Expressão e caracterização farmacológica dos subtipos de adrenoceptores α1 na cauda proximal e distal do epidídimo de rato
(Universidade Estadual Paulista (Unesp), 2012-06-12)
O epidídimo é um órgão formado por um longo túbulo enovelado composto por 3 regiões anatômicas distintas: a cabeça, o corpo e a cauda. A cabeça e o corpo do epidídimo têm papel na maturação dos espermatozóides, enquanto ...
Expressão e caracterização farmacológica dos subtipos de adrenoceptores α1 na cauda proximal e distal do epidídimo de rato
(Universidade Estadual Paulista (Unesp), 2012-06-12)
O epidídimo é um órgão formado por um longo túbulo enovelado composto por 3 regiões anatômicas distintas: a cabeça, o corpo e a cauda. A cabeça e o corpo do epidídimo têm papel na maturação dos espermatozóides, enquanto ...
Evaluation of benzyltetrahydroisoquinolines as ligands for neuronal nicotinic acetylcholine receptors
(Nature Publishing Group, 2005-06-27)
1 Effects of derivatives of coclaurine (C), which mimic the ‘eastern’ or the nonquaternary halves of
the alkaloids tetrandrine or d-tubocurarine, respectively, both of which are inhibitors of nicotinic
acetylcholine ...