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Synthesis, Antifungal and Antitumor Activity of Novel (Z)-5-Hetarylmethylidene-1,3-thiazol-4-ones and (Z)-5-Ethylidene-1,3-thiazol-4-ones
(Universidad del Rosario, 2013)
New hetaryl- and alkylidenerhodanine derivatives 3a-d, 3e, and 4a-d were prepared from heterocyclic aldehydes 1a-d or acetaldehyde 1e. The treatment of several rhodanine derivatives 3a-d and 3e with piperidine or morpholine ...
(e)-2-(benzo[d]thiazol-2-yl)-3-heteroarylacrylonitriles as efficient michael acceptors for cysteine: real application in biological imaging
(ELSEVIER SCIENCE SA, 2014)
(E)-2-(Benzo[d]thiazol-2-yl)-3-heteroarylacrylonitriles derivatives (compounds 1, 2, and 3) were synthesized and assessed for their ability to recognize cysteine (Cys) in aqueous solution via a Michael-type reaction. The ...
Synthesis of novel thiazole-based 8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepines as potential antitumor and antifungal agents
(Elsevier Masson, 2015-03)
A new series of novel thiazole-based 8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepines 6a–g and 7a–g were obtained with high regioselectivity from the reaction of triamino- or tetraaminopyrimidines 4 and 5 with α,β-unsaturated ...
Crystal structure of 2-fluoro-N-(1,3-thiazol-2-yl)benzamide
(2015-10-24)
In the title compound, C10H7FN2OS, the mean plane of the
central amide fragment (r.m.s. deviation = 0.048 A˚ ) makes
dihedral angles of 35.28 (8) and 10.14 (12) with those of the
fluorobenzene and thiazole rings, ...
Anti-liver cancer activity in vitro and in vivo induced by 2-pyridyl 2,3-thiazole derivatives
(Brasil, 2018-05-04)
A total of 24 hybrid compounds containing pyridyl and 1,3-thiazole moieties were screened against HL-60 (leukemia),
MCF-7 (breast adenocarcinoma),HepG2 (hepatocellular carcinoma), NCI-H292 (lung carcinoma) human
tumor cell ...