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Avaliação das propriedades antitumorais de complexos de rutênio(II) contendo os ligantes lapachol ou lausona
(Universidade Federal de São CarlosUFSCarPrograma de Pós-Graduação em Química - PPGQCâmpus São Carlos, 2018-06-29)
Metal complexes containing ligands that present biological activity have been attracting interest in the field of development of new drugs for the treatment of cancer. Lapachol and lawsone are examples of important natural ...
Atividade antimicrobiana "in vitro" e determinação da concentração inibitória mínina (CIM) de fitoconstituintes e produtos sintéticos sobre bactérias e fungos leveduriformes
(2006)
Diante da problemática da resistência microbiana as pesquisas apontam para o uso de novos antibióticos que sejam eficazes ante os patógenos emergentes. Este trabalho objetiva testar frente a bactérias gram-positivas ...
Antiparasitic activities of novel ruthenium/lapachol complexes
(ElsevierPhiladelphia, 2014-07)
The present study describes the synthesis, characterization, antileishmanial and antiplasmodial activities of novel diimine/(2,2′-bipyridine (bipy), 1,10-phenanthroline (phen), 4,4′-methylbipyridine (Me-bipy) and 4,4′- ...
Preparación de derivados 1,2,3-triazol-lapachol vía click chemistry
(Universidad de Talca (Chile). Escuela de Tecnología Médica., 2018)
Síntesis de nuevos derivados triazol-lapachol mediante reacción de cicloadición 1,3-dipolar
(Universidad de Talca (Chile). Escuela de Tecnología Médica., 2018)
Natural and synthetic naphthoquinones active against Trypanosoma cruzi: An initial step towards new drugs for chagas disease
(2011)
Chagas disease is one of the most important endemic diseases in Latin America, caused by Trypanosoma cruzi. The drugs used for the treatment of this disease, nifurtimox and benznidazole, are toxic and present severe side ...
Isolation of Major Components from the Roots of Godmania aesculifolia and Determination of Their Antifungal Activities
(2013)
From the methanol root extract of Godmania aesculifolia, a species selected in a multinational OAS program aimed at discovering antifungal compounds from Latin American plants, a new chavicol diglycoside (1), the known ...
Spasmolytic activity of lapachol and its derivatives, α and β-lapachone, on the guinea-pig ileum involves blockade of voltage-gated calcium channels
(2008)
O lapachol, α e β-lapachona são naftoquinonas obtidas de espécies de Tabebuia, apresentam propriedades antiinflamatória, antibacteriana, anticâncer e tripanossomicida. O objetivo deste trabalho foi investigar um possível ...