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Avaliação do potencial antitumoral in vitro dos derivados sintéticos do indolEvaluation of the in vitro antitumoral potential of indol synthetic derivatives
(Pós-Graduação em Ciências FisiológicasUniversidade Federal de Sergipe (UFS), 2023)
Effects of indole alkaloids from gramineae on aphids
(1984)
The indole bases N∞-methyltryptamine, 5-methoxy-N, N-dimethyltryptamine, 3-N,N-dimethylaminomethylindole (gramine) and 5-methoxytryptamine decreased survival of nymphs of Rhopalosiphum maidis with LD50 of 3.8, 3.5, 2.9 and ...
Synthesis and preliminary evaluation of 3-thiocyanato-1H-indoles as potential anticancer agents
(Elsevier France-editions Scientifiques Medicales Elsevier, 2016-08)
A novel series of twenty 3-thiocyanato-1H-indoles, carrying diversification at positions N-1, C-2 and C-5 of the heterocyclic core, were synthesized; their antiproliferative activity against four human cancer cell lines ...
Estudio de síntesis de arilpiperazinilacetilpiperazinil-propil-1h-indoles como potenciales ligandos de acción multireceptorial
(Universidad de Chile, 2016)
El presente trabajo de memoria informa sobre la preparación de dos familias de
derivados indólicos polifuncionalizados: 3-(3-{4-[(aril-1-piperazinil)acetil]-1-piperazinil}propil)-
1H-indoles (Familia I) y 5-fluoro-3-(3 ...
Síntese, caracterização e avaliação antitumoral de novos derivados 3-Benzil-5-(Indol-3-il-Metileno)-Tiazolidina-2,4-Diona
(Universidade Federal de Pernambuco, 2014)
New synthetic method of N-indol-glycosides with antimicrobial activity
(Sociedad Chilena De QuimicaConcepcionChile, 1998)
Síntese de 3-iodo-4H-calcogenofeno[3,2-b]indol via ciclização eletrofílica mediada por iodo de derivados de alquinil indol
(Universidade Federal de Santa MariaBrasilQuímicaUFSMPrograma de Pós-Graduação em QuímicaCentro de Ciências Naturais e Exatas, 2019-07-26)
The treatment of alkynyl índoles by using iodine with electrophilic source led to 3-iodo-4H-calcogenophene[3,2-b]indoles derivates. Firstly a series of studies were performed variations to obtain the compounds containing ...
Indole-3-carbaldehyde semicarbazone derivatives: synthesis, characterization, and antibacterial activities
(Hindawi, 2020)
Four indole-3-carbaldehyde semicarbazone derivatives, 2-((5-bromo-1H-indol-3-yl)methylene)hydrazinecarboxamide (1), 2-((5-chloro-1H-indol-3-yl)methylene)hydrazinecarboxamide (2), 2-((5-methoxy-1H-indol-3-yl)methylene)hyd ...
Pd-Catalyzed alfa-Arylation of Sulfones in a Three-Component Synthesis 3-[2-(phenyl/methylsulfonyl)ethyl]indoles
(American Chemical Society, 2016-02)
A novel four-step domino process for the synthesis of 3-[2-(aryl/alkylsulfonyl)ethyl]indoles starting from readily available 2-iodoanilines is reported. The domino reaction is based on the intramolecular palladium-catalyzed ...
Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis
(2017-01-01)
The neuroleptic drug thioridazine has been recently repositioned as possible anti-tubercular drug. Thioridazine showed anti-tubercular activity against drug resistant mycobacteria but it is endowed with adverse side effects. ...