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Produtos naturais como candidatos a fármacos úteis no tratamento do mal de Alzheimer
(2004-07-01)
Alzheimer's disease (AD) is a progressive neurodegenerative pathology with severe economic and social impact. There is currently no cure, although cholinesterase inhibitors provide effective temporary relief of symptoms ...
A synopsis on the linkage between age-related dementias and vascular disorders
(Bentham Science Publishers B.V., 2016)
Design, Synthesis, Biological Evaluation and Molecular Modelling of Substituted pyrrolo[2,1-a]isoquinolinone derivatives: Discovery of Potent Inhibitors of AChE and BChE
(Royal Society of Chemistry, 2021-04)
We report here the design, synthesis and biological evaluation of a new series of substituted pyrrolo[2,1-a]isoquinolin-3-one derivatives, some of which have strong inhibitory activity against both AChE and BChE enzymes. ...
Encapsulamento de rivastigmina em nanopartículas de P(MMA-co-AA) funcionalizadas para tratamento de doenças neurodegenerativas
(Universidade Federal do Rio de JaneiroBrasilInstituto Alberto Luiz Coimbra de Pós-Graduação e Pesquisa de EngenhariaPrograma de Pós-Graduação em Engenharia QuímicaUFRJ, 2020)
Cholinesterase inhibitors effects in patients with Lewy's bodies associated diseaseEfectos de inhibidores de colinesterasa en pacientes con enfermedad asociada a cuerpos de Lewy
(Universidad Nacional Mayor de San Marcos, Facultad de Medicina Humana, 2008)
Determinación en membranas celulares y modelos moleculares del efecto protector de drogas utilizadas en la enfermedad de Alzheimer.Determination in cell membranes and molecular models of the protective effect of drugs used in Alzheimer's disease.
(2019)
El péptido beta amiloide (Aβ) es tóxico para las neuronas. Desde hace más de una década se han examinado los efectos de medicamentos que tienen una acción inhibidora de la acetilcolinesterasa, con lo cual se han mejorado ...
Neuropsychiatric symptoms related to cholinergic deficits in Parkinson’s disease
(Springer Nature, 2017)
Abstract: Given its ability to explain the most frequent motor symptoms of Parkinson’s disease (PD), degeneration of dopaminergic neurons has been considered one of the disease´s main pathophysiological features. Several ...