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Reaction of 4,5-diamino-3-methyl-1-phenylpyrazole with 3-dimethylaminopropiophenones. Synthesis of new 4-aryl-6-methyl-8-phenyl-2,3-dihydropyrazolo[3,4-b]diazepines and 4-aryl-8-methyl-6-phenyl-2,3-dihydropyrazolo[4,3-b]diazepines
(HETERO CORPORATION, 1999-05)
New 4-Aryl-6-methyl-8-phenyl-2,3-dihydropyrazolo[3,4-b]diazepines and 4-aryl-8-methyl-6-phenyl-2,3-dihydropyrazolo[4,3-b]diazepines were obtained from the reaction of 4,5-diamino-3-methyl-1-phenylpyrazole 1 with one ...
Reaction of 4,5-diamino-3-methyl-1-phenylpyrazole with 3- dimethylaminopropiophenones. Synthesis of new 4-aryl-6-methyl-8-phenyl-2,3- dihydropyrazolo[3,4-b]diazepines and 4-aryl-8-methyl-6-phenyl-2,3- dihydropyrazolo[4,3-b]diazepines
(HeteroCorporation, 1999)
New 4-Aryl-6-methyl-8-phenyl-2,3-dihydropyrazolo[3,4-b]diazepines and 4- aryl-8-methyl-6-phenyl-2,3-dihydropyrazolo[4,3-b]diazepines were obtained from the reaction of 4,5-diamino-3-methyl-1-phenylpyrazole 1 with one ...
Synthesis of new 1-benzyl-4,6-diaryl-2,3-dihydropyrazolo[3,4-b][1,4]diazepines
(FREUND PUBLISHING HOUSE LTD, 2000)
The reaction of 4-amino-3-aryl-5-benzylaminopyrazoles (1a,b) with 3-dimethylaminopropiophenones (2) in ethanol with acetic acid gave 1-benzyl-4,6-diaryl-2,3-dihydropyrazolo[3,4-b] [1,4]diazepines (3a-h). The structure ...
Enol-imino-keto-enamine tautomerism in a diazepine derivative: How decisive are the intermolecular interactions in the equilibrium?
(American Chemical Society, 2019-08)
The strange tautomeric equilibrium behaviour exhibited by a new o-hydroxyphenyl diazepine derivative, when the compound is analysed both in solution and solid state, open the structural study of the enol-imino-keto-enamine ...
Synthesis of novel thiazole-based 8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepines as potential antitumor and antifungal agents
(Elsevier Masson, 2015-03)
A new series of novel thiazole-based 8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepines 6a–g and 7a–g were obtained with high regioselectivity from the reaction of triamino- or tetraaminopyrimidines 4 and 5 with α,β-unsaturated ...
Reaction of 4,5,6-triaminopyrimidine and 2,4,5,6-tetraaminopyrimidine with 3-dimethylaminopropiophenones. Synthesis of new 4-aryl-2,3- dihydropyrimido[4,5-b][1,4]diazepines
(HeteroCorporation, 2000)
Several new 6-amino- and 6,8-diamino-4-aryl-2,3-dihydropyrimido[4,5- b][1,4]diazepines were obtained from the reaction of 4,5,6-triaminopyrimidine 1a and 2,4,5,6-tetraaminopyrimidine 1b with one equivalent of 3- ...
Reaction of 4,5,6-triaminopyrimidine and 2,4,5,6-tetraaminopyrimidine with 3-dimethylaminopropiophenones. Synthesis of new 4-aryl-2,3-dihydropyrimido[4,5-b][1,4]diazepines
(HETERO CORPORATION, 2000-03)
Several new 6-amino- and 6,8-dinmino-4-aryl-2,3-dihydropyrimido[4,5-b][1,4]diazepines were obtained from the reaction of 4,5,6-triaminopyrimidine 1a and 2,4,5,6-tetraaminopyrimidine 1b with one equivalent of 3-dimethylam ...
1,n-Diamines. Part 3: Microwave-assisted synthesis of N-acyl-N′-arylhexahydropyrimidines and hexahydro-1,3-diazepines
(Pergamon-Elsevier Science Ltd, 2011-10)
In this Letter we present a method for the synthesis of N-acyl-N´-arylhexahydropyrimidines 1, by ring closure of N-acyl-N´-aryl-1,3-propanediamines 3 with formaldehyde. Cyclodehydrations were performed in aqueous medium ...